Question: Moving to the next question prevents changes to this answer. uestion 5 Which of the following is not true of Transition-State Inhibitors? a. Thy bind

Moving to the next question prevents changes to this answer. uestion 5 Which of the following is not true of Transition-State Inhibitors? a. Thy bind more strongly to the active site than drugs that mimic the substrate or product. b. They react reversibly with the enzyme by non-covalent interactions. c. They mimics the stereochemistry of the transition state of an enzyme-catalysed reaction, but they are not stable. d. They are so called because they mimic the transition state of an enzyme-catalysed reaction Lrestion 6 Which of the following is required to achieve an efficient competitive enzyme inhibition? a. A drug should form stronger non-covalent interactions with active site compared to the substrate. b. A drug should bind to the active site to be converted to an electrophilic product c. A drug should form a strong covalent bond with the active site. d. A drug should have higher concentration than the substrate e. Both a and d
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